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Structure–activity relationship study of novel tissue transglutaminase inhibitors

Eric Duval, April Case, Ross L. Stein, Gregory D. Cuny

Bioorganic & Medicinal Chemistry Letters · 2005 · 89 citations · 10 references

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10

Identification of tissue transglutaminase as the autoantigen of celiac disease

Walburga Dieterich, Tobias Ehnis, Michael Bauer et al. · Nature Medicine · 1997 · 2.1K citations

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‘Tissue’ transglutaminase ablation reduces neuronal death and prolongs survival in a mouse model of Huntington's disease

Pier G. Mastroberardino, Carlo Iannicola, Roberta Nardacci et al. · Cell Death and Differentiation · 2002 · 227 citations · Full text

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Thiophene systems. 9. Thienopyrimidinedione derivatives as potential antihypertensive agents

Ronald K. Russell, Jeffery B. Press, Richard Rampulla et al. · Journal of Medicinal Chemistry · 1988 · 179 citations · Full text

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Discovery of a Thieno[2,3- <i>d</i> ]pyrimidine-2,4-dione Bearing a <i>p</i> -Methoxyureidophenyl Moiety at the 6-Position:  A Highly Potent and Orally Bioavailable Non-Peptide Antagonist for the Human Luteinizing Hormone-Releasing Hormone Receptor

Satoshi Sasaki, Nobuo Cho, Yoshi Nara et al. · Journal of Medicinal Chemistry · 2002 · 161 citations · Full text

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Discovery and SAR of a Novel Selective and Orally Bioavailable Nonpeptide Classical Competitive Inhibitor Class of Protein-Tyrosine Phosphatase 1B

Henrik Sune Andersen, Ole H. Olsen, Lars Iversen et al. · Journal of Medicinal Chemistry · 2002 · 133 citations · Full text

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