Publication | Closed Access

Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism

Structural CharacterizationSignal TransductionFunctional SelectivityG Protein-coupled ReceptorHormonal ReceptorReceptor (Biochemistry)Molecular BiologyEstrogen Receptor AntagonismNon-peptide LigandSubtype-selective LigandEndocrinologyMedicineBiomolecular EngineeringDrug Discovery