Publication | Open Access

Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-(2-(4′-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine (APD916)

Histamine H3 ReceptorMolecular PharmacologyMedicinal ChemistryBiochemistryMedicineNatural SciencesMechanism Of ActionBiaryl Sulfone DerivativesPharmacological AgentReceptor (Biochemistry)PharmacotherapyPharmacologyPharmaceutical ChemistryDrug Discovery