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Binding Characteristics of Cetirizine and Levocetirizine to Human H<sub>1</sub>Histamine Receptors: Contribution of Lys<sup>191</sup>and Thr<sup>194</sup>

Michel Gillard, Christy Van Der Perren, Nicole Moguilevsky, R. Massingham, Pierre Chatelain

Molecular Pharmacology · 2002 · 210 citations · 21 references

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References

21

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.8K citations

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Cloning and Functional Expression of the Human Histamine H<sub>3</sub>Receptor

Timothy W. Lovenberg, Barbara Roland, Sandy J. Wilson et al. · Molecular Pharmacology · 1999 · 700 citations · Full text

Molecular Cloning and Characterization of a Novel Type of Histamine Receptor Preferentially Expressed in Leukocytes

Tamaki Oda, Noriyuki Morikawa, Yoko Saito et al. · Journal of Biological Chemistry · 2000 · 610 citations · Full text

Validation and statistical analysis of a computer modeling method for quantitative analysis of radioligand binding data for mixtures of pharmacological receptor subtypes.

A. De Léan, Arthur A. Hancock, Robert J. Lefkowitz · Molecular Pharmacology · 1982 · 594 citations

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The kinetics of competitive radioligand binding predicted by the law of mass action.

Harvey Motulsky, L C Mahan · Molecular Pharmacology · 1984 · 417 citations