Comparison of Pharmacological Activities of Buprenorphine and Norbuprenorphine: Norbuprenorphine Is a Potent Opioid Agonist

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Orphanin FQ: A Neuropeptide That Activates an Opioidlike G Protein-Coupled Receptor

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Cloning of a Delta Opioid Receptor by Functional Expression

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A practical computer-based approach to the analysis of radioligand binding experiments

Grant A. McPherson · Computer Programs in Biomedicine · 1983 · 832 citations

Pharmacy, Biochemistry, Chemistry +10