Concepedia

Identification, synthesis, and biological evaluation of novel pyrazoles as low molecular weight luteinizing hormone receptor agonists

Catherine Jorand‐Lebrun, Bill Brondyk, Jing‐Jer Lin, Sharad S. Magar, Robert Murray, Adulla Reddy, Hitesh N. Shroff, Greg Wands, W Y Weiser, Qihong Xu,

Bioorganic & Medicinal Chemistry Letters · 2006 · 40 citations · 6 references

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References

6

Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors:  Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1<i>H</i>-pyrazol-1-yl]benzenesulfonamide (SC-58635, Celecoxib)

Thomas D. Penning, John J. Talley, Stephen R. Bertenshaw et al. · Journal of Medicinal Chemistry · 1997 · 2K citations · Full text

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Structural predictions for the ligand-binding region of glycoprotein hormone receptors and the nature of hormone–receptor interactions

Xuliang Jiang, Michel Dréano, David R. Buckler et al. · Structure · 1995 · 188 citations · Full text

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The First Orally Active Low Molecular Weight Agonists for the LH Receptor: Thienopyr(im)idines with Therapeutic Potential for Ovulation Induction

Nicole C.R. van Straten, G. G. Schoonus-Gerritsma, R. G. van Someren et al. · ChemBioChem · 2002 · 104 citations

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Estrogen pyrazoles: defining the pyrazole core structure and the orientation of substituents in the ligand binding pocket of the estrogen receptor

Shaun R. Stauffer, Ying Huang, Christopher J. Coletta et al. · Bioorganic & Medicinal Chemistry · 2001 · 92 citations

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Identification of Substituted 6-Amino-4-phenyltetrahydroquinoline Derivatives:  Potent Antagonists for the Follicle-Stimulating Hormone Receptor

Nicole C.R. van Straten, Twan H. J. van Berkel, Dennis Demont et al. · Journal of Medicinal Chemistry · 2004 · 81 citations · Full text

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