Regioselective reactivity of some 5,7-dimethoxyindoles

Efficient Reagents for the Synthesis of 5-, 7-, and 5,7-Substituted Indoles Starting from Aromatic Amines:  Scope and Limitations

Jesús Ezquerra, Concepción Pedregal, Carlos José Einicker Lamas et al. · The Journal of Organic Chemistry · 1996 · 186 citations

Natural Sciences, Chemistry, Medicinal Chemistry +13

Duocarmycin-pyrindamycin DNA alkylation properties and identification, synthesis, and evaluation of agents incorporating the pharmacophore of the duocarmycin-pyrindamycin alkylation subunit. Identification of the CC-1065 duocarmycin common pharmacophore

Dale L. Boger, Takayoshi Ishizaki, Hamideh Zarrinmayeh et al. · Journal of the American Chemical Society · 1990 · 136 citations

Medicine, Medicinal Chemistry, Pharmacology +7

Entry into 6-Methoxy-D(+)-tryptophans. Stereospecific Synthesis of 1-Benzenesulfonyl-6-methoxy-D(+)-tryptophan Ethyl Ester

M.S. Allen, Linda K. Hamaker, Anthony J. La Loggia et al. · Synthetic Communications · 1992 · 69 citations

Natural Sciences, Chemistry, Medicinal Chemistry +12

Substitution, oxidation and addition reactions at C-7 of activated indoles

D. ST. C. BLACK, Michael C. Bowyer, Maria M. Catalano et al. · Tetrahedron · 1994 · 56 citations

Natural Sciences, Chemistry, Organic Chemistry +11

Synthesis of Activated 3-Arylindoles

DS Black, MC Bowyer, P. M. Bowyer et al. · Australian Journal of Chemistry · 1994 · 45 citations

Natural Sciences, Chemistry, Medicinal Chemistry +8