SLAS DISCOVERY · 2006 · 35 citations · 18 references
PharmacyMedicinal ChemistryMolecular BiologyDrug DesignDrug DiscoveryMass Spectrometric AnalysisDrug-target Interaction MappingHigh-throughput ScreeningMolecular ScreeningProtein-ligand RecognitionSmall-molecule ScreeningAffinity ScreeningAffinity SelectionAffinity Selection-mass SpectrometryCheckpoint Kinase InhibitionKinase Binding AssaysKinase InhibitorsMass Spectral Data AnalysisMass Spectrometry-based Screening
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Specificity and mechanism of action of some commonly used protein kinase inhibitors
Stephen Davies, Helen Reddy, Matilde Caivano et al. · Biochemical Journal · 2000 · 4.1K citations · Full text
Specificity and mechanism of action of some commonly used protein kinase inhibitors
Stephen Davies, Helen Reddy, Matilde Caivano et al. · Biochemical Journal · 2000 · 3.1K citations
Structural Mechanism for STI-571 Inhibition of Abelson Tyrosine Kinase
Thomas H. Schindler, William G. Bornmann, Patricia Pellicena et al. · Science · 2000 · 1.8K citations