The Identification of a Novel Phosphodiesterase 4 Inhibitor, 1-Ethyl-5-{5-[(4-methyl-1-piperazinyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-b]pyridin-4-amine (EPPA-1), with Improved Therapeutic Index using Pica Feeding in Rats as a Measure of Emetogenicity

Trong Davis, John J. Peterson, Jen-Pyng Kou, Elizabeth A. Capper-Spudich, D.I. Ball, Anthony T. Nials, Joanne Wiseman, Yemisi Solanke, Fiona S. Lucas, Richard A. Williamson,

Journal of Pharmacology and Experimental Therapeutics · 2009 · 21 citations · 22 references

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