Concepedia

Multiple Differences in Agonist and Antagonist Pharmacology between Human and Guinea Pig Histamine H1-Receptor

Roland Seifert, Katharina Wenzel‐Seifert, Tilmann Bürckstümmer, Heinz H. Pertz, Walter Schunack, Stefan Dove, Armin Buschauer, Sigurd Elz

Journal of Pharmacology and Experimental Therapeutics · 2003 · 79 citations · 36 references

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References

36

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Crystal Structure of Rhodopsin: A G Protein-Coupled Receptor

Krzysztof Palczewski, Takashi Kumasaka, Tetsuya Hori et al. · Science · 2000 · 5.6K citations

, , +16

Structural Mimicry in G Protein-Coupled Receptors: Implications of the High-Resolution Structure of Rhodopsin for Structure-Function Analysis of Rhodopsin-Like Receptors

Juan Antonio Ballesteros‐Cánovas, Lei Shi, Jonathan A. Javitch · Molecular Pharmacology · 2001 · 440 citations

, , +17

Genomics Meets Histamine Receptors: New Subtypes, New Receptors

Lindsay B. Hough · Molecular Pharmacology · 2001 · 311 citations

, , +12

Histamine H<sub>1</sub>-Receptor Activation of Nuclear Factor-κB: Roles for Gβγ- and Gα<sub>q/11</sub>-Subunits in Constitutive and Agonist-Mediated Signaling

Remko A. Bakker, Stefan B. J. Schoonus, Martine J. Smit et al. · Molecular Pharmacology · 2001 · 258 citations

, , +14