Concepedia

A Novel Phenylaminotetralin Radioligand Reveals a Subpopulation of Histamine H1 Receptors

Raymond G. Booth, Nader H. Moniri, Remko A. Bakker, Neepa Choksi, William B. Nix, Henk Timmerman, Rob Leurs

Journal of Pharmacology and Experimental Therapeutics · 2002 · 23 citations · 32 references

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References

32

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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A ternary complex model explains the agonist-specific binding properties of the adenylate cyclase-coupled beta-adrenergic receptor.

A. De Léan, Jeffrey M. Stadel, Robert J. Lefkowitz · Journal of Biological Chemistry · 1980 · 1.6K citations · Full text

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A Peptide Derived from a β2-Adrenergic Receptor Transmembrane Domain Inhibits Both Receptor Dimerization and Activation

Terence E. Hébert, Serge Moffett, Jean-Pierre Morello et al. · Journal of Biological Chemistry · 1996 · 770 citations · Full text

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Dimerization of the δ Opioid Receptor:

Svetlana Cvejic, Lakshmi A. Devi · Journal of Biological Chemistry · 1997 · 482 citations · Full text

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Histamine H<sub>1</sub>-Receptor Activation of Nuclear Factor-κB: Roles for Gβγ- and Gα<sub>q/11</sub>-Subunits in Constitutive and Agonist-Mediated Signaling

Remko A. Bakker, Stefan B. J. Schoonus, Martine J. Smit et al. · Molecular Pharmacology · 2001 · 258 citations

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