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Synthesis of benzamide derivatives as TRPV1 antagonists

Yuji Shishido, Madoka Jinno, Takafumi Ikeda, Fumitaka Ito, Masaki Sudo, Naoya Makita, Atsuko Ohta, Ayako Iki-Taki, Takashi Ohmi, Yoshihito Kanai,

Bioorganic & Medicinal Chemistry Letters · 2007 · 18 citations · 12 references

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12

The capsaicin receptor: a heat-activated ion channel in the pain pathway

Michael J. Caterina, Mark Schumacher, Makoto Tominaga et al. · Nature · 1997 · 9.1K citations

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Impaired Nociception and Pain Sensation in Mice Lacking the Capsaicin Receptor

Michael J. Caterina, Andreas Leffler, Annika B. Malmberg et al. · Science · 2000 · 3.5K citations

, , +17

The Cloned Capsaicin Receptor Integrates Multiple Pain-Producing Stimuli

Makoto Tominaga, Michael J. Caterina, Annika B. Malmberg et al. · Neuron · 1998 · 3.1K citations · Full text

, , +14

Vanilloid receptor-1 is essential for inflammatory thermal hyperalgesia

John B. Davis, Julie Gray, Martin J. Gunthorpe et al. · Nature · 2000 · 1.8K citations

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Capsazepine: a competitive antagonist of the sensory neurone excitant capsaicin

Stuart Bevan, Sandeep S Hothi, Glyn A. Hughes et al. · British Journal of Pharmacology · 1992 · 584 citations · Full text

, , +16