Concepedia

Cloning of Rat Histamine H3 Receptor Reveals Distinct Species Pharmacological Profiles

Timothy W. Lovenberg, Jayashree Pyati, Hong Chang, Sandy J. Wilson, Mark G. Erlander

Journal of Pharmacology and Experimental Therapeutics · 2000 · 187 citations · 25 references

Open access

Concepts

MedicineNeurobiologyPharmacologyCell SignalingMolecular PharmacologyNeuropharmacologyNeurotransmissionReceptor PharmacologyReceptor PhysiologyAgonist ActivityAntagonist ActivityAntagonist PotencyCloningHistamine Receptor AntagonistsHistamine Receptor PharmacologyHistamine Receptors

References

25

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

Life Sciences, Biochemistry, Chemical Kinetics +14

Rapid and Sensitive Protein Similarity Searches

David J. Lipman, William R. Pearson · Science · 1985 · 4.1K citations

Life Sciences, Bioinformatics, Molecular Biology +16

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

Life Sciences, Neuroscience, Pharmacology +14

Cloning and Functional Expression of the Human Histamine H<sub>3</sub>Receptor

Timothy W. Lovenberg, Barbara Roland, Sandy J. Wilson et al. · Molecular Pharmacology · 1999 · 700 citations · Full text

Life Sciences, Neuroscience, Pharmacology +16

pA<sub>x</sub> AND COMPETITIVE DRUG ANTAGONISM

H. O. Schild · British Journal of Pharmacology and Chemotherapy · 1949 · 245 citations · Full text

Medicine, Pharmacology, Experimental Pharmacology +10