Concepedia

Inhibition of secretory phospholipase A. 1-Design, synthesis and structure–activity relationship studies starting from 4-tetradecyloxybenzamidine to obtain specific inhibitors of group II sPLAs

Leon Assogba, Azali Ahamada‐Himidi, Nadia Meddad-Bel Habich, Darina Aoun, Latifa Boukli, France Massicot, Carine M. Mounier, Jack Huet, Aazdine Lamouri, Jean‐Edouard Ombetta

European Journal of Medicinal Chemistry · 2005 · 19 citations · 19 references

DOI

Concepts

References

19

Induction of phospholipase A2 gene expression in human hepatoma cells by mediators of the acute phase response

Robert M. Crowl, T J Stoller, Robert R. Conroy et al. · Journal of Biological Chemistry · 1991 · 408 citations · Full text

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Synthesis and Angiotensin II Receptor Antagonistic Activities of Benzimidazole Derivatives Bearing Acidic Heterocycles as Novel Tetrazole Bioisosteres

Yasuhisa Kohara, Keiji Kubo, Eiko Imamiya et al. · Journal of Medicinal Chemistry · 1996 · 272 citations

, , +16

Structures of Free and Inhibited Human Secretory Phospholipase A <sub>2</sub> from Inflammatory Exudate

David L. Scott, Steven P. White, Jeffrey L. Browning et al. · Science · 1991 · 252 citations

, , +16

Structure of recombinant human rheumatoid arthritic synovial fluid phospholipase A2 at 2.2 Å resolution

Jean‐Pierre Wery, Richard W. Schevitz, David K. Clawson et al. · Nature · 1991 · 201 citations

, , +10

Novel 1,2,4-oxadiazoles and 1,2,4-thiadiazoles as dual 5-lipoxygenase and cyclooxygenase inhibitors

Paul C. Unangst, G. P. SHRUM, D. T. CONNOR et al. · Journal of Medicinal Chemistry · 1992 · 198 citations · Full text

, , +9