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The influence of modifications in imide fragment structure on 5-HT1A and 5-HT7 receptor affinity and in vivo pharmacological properties of some new 1-(m-trifluoromethylphenyl)piperazines

Maria H. Paluchowska, Ryszard Bugno, Beata Duszyńska, E Tatarczyńska, Agnieszka Nikiforuk, Tomasz Lenda, E Chojnacka-Wójcik

Bioorganic & Medicinal Chemistry · 2007 · 57 citations · 27 references

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References

27

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

A pharmacological profile of the selective silent 5-HT1A receptor antagonist, WAY-100635

Elaine A. Forster, Ian A. Cliffe, David J. Bill et al. · European Journal of Pharmacology · 1995 · 611 citations

, , +8

The pharmacology of the hypothermic response in mice to 8-hydroxy-2-(DI-n-propylamino)tetralin (8-OH-DPAT)

Guy M. Goodwin, R.J. De Souza, A.R. Green · Neuropharmacology · 1985 · 254 citations

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Effect of the selective 5-HT7 receptor antagonist SB 269970 in animal models of anxiety and depression

Anna Wesołowska, Agnieszka Nikiforuk, Katarzyna Stachowicz et al. · Neuropharmacology · 2006 · 227 citations

, , +12

Evaluation of a rapid technique for detecting minor tranquilizers

C Aron, Pierre Simon, C Larousse et al. · Neuropharmacology · 1971 · 171 citations

, , +2