Metabolic stability of 6,7-dialkoxy-4-(2-, 3- and 4-[18F]fluoroanilino)quinazolines, potential EGFR imaging probes

A Specific Inhibitor of the Epidermal Growth Factor Receptor Tyrosine Kinase

David W. Fry, Alan J. Kraker, Amy McMichael et al. · Science · 1994 · 802 citations

Life Sciences, Oncology, Pharmacology +15

Tyrosine Kinase Inhibitors. 8. An Unusually Steep Structure−Activity Relationship for Analogues of 4-(3-Bromoanilino)-6,7-dimethoxyquinazoline (PD 153035), a Potent Inhibitor of the Epidermal Growth Factor Receptor

Alexander J. Bridges, Hairong Zhou, Donna R. Cody et al. · Journal of Medicinal Chemistry · 1996 · 322 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Aryltrimethylammonium trifluoromethanesulfonates as precursors to aryl [¹⁸F]fluorides: Improved synthesis of [¹⁸F]GBR‐13119

Michael Haka, Michael R. Kilbourn, G. Leonard Watkins et al. · Journal of Labelled Compounds and Radiopharmaceuticals · 1989 · 180 citations

Natural Sciences, Chemistry, Medicinal Chemistry +10

Potential 18F-labeled biomarkers for epidermal growth factor receptor tyrosine kinase

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Life Sciences, Biochemistry, Molecular Biology +11

Labeled aryl fluorides from the nucleophilic displacement of activated nitro groups by ¹⁸F‐F⁻

Marina Attinà, Fulvio Cacace, Alfred P. Wolf · Journal of Labelled Compounds and Radiopharmaceuticals · 1983 · 74 citations

Natural Sciences, Chemistry, Analytical Chemistry +9