Concepedia

Potent dual antagonists of endothelin and angiotensin II receptors derived from α-phenoxyphenylacetic acids (Part III)

Thomas F. Walsh, Kenneth J. Fitch, David L. Williams, Kathryn L. Murphy, Nancy A. Nolan, Douglas J. Pettibone, Raymond S.L. Chang, Stacey O’Malley, Bradley V. Clineschmidt, Daniel F. Veber,

Bioorganic & Medicinal Chemistry Letters · 1995 · 35 citations · 14 references

DOI

Concepts

References

14

Cloning and expression of a cDNA encoding an endothelin receptor

Hiroshi Arai, Seiji Hori, Ichiro Aramori et al. · Nature · 1990 · 2.6K citations

, , +7

Cloning of a cDNA encoding a non-isopeptide-selective subtype of the endothelin receptor

Takeshi Sakurai, Masashi Yanagisawa, Yoh Takuwat et al. · Nature · 1990 · 2.4K citations · Full text

, , +8

Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor

Masaki Ihara, Kazuhito Noguchi, Toshihiko Saeki et al. · Life Sciences · 1992 · 877 citations

, , +7

Pathophysiological role of endothelin revealed by the first orally active endothelin receptor antagonist

Martine Clozel, Volker Breu, Kaspar F. Burri et al. · Nature · 1993 · 529 citations

, , +9

The endothelin ETB receptor mediates both vasodilation and vasoconstriction in vivo

Martine Clozel, Gillian A. Gray, Volker Breu et al. · Biochemical and Biophysical Research Communications · 1992 · 402 citations

, , +9