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Expanding the repertoire of small molecule transcriptional activation domains

Ryan Casey, Jean‐Paul Desaulniers, Jonas W. Højfeldt, Anna K. Mapp

Bioorganic & Medicinal Chemistry · 2008 · 12 citations · 22 references

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References

22

Solution Structure of the KIX Domain of CBP Bound to the Transactivation Domain of CREB: A Model for Activator:Coactivator Interactions

Ishwar Radhakrishnan, Gabriela C. Pérez-Alvarado, David Parker et al. · Cell · 1997 · 730 citations · Full text

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Induced α Helix in the VP16 Activation Domain upon Binding to a Human TAF

Motonari Uesugi, Origène Nyanguile, Hua Lu et al. · Science · 1997 · 290 citations

, , +17

Generating yeast transcriptional activators containing no yeast protein sequences

Douglas M. Ruden, Jun Ma, Yi Li et al. · Nature · 1991 · 177 citations

, , +13

Structural Basis for Cooperative Transcription Factor Binding to the CBP Coactivator

Roberto N. De Guzman, Natalie K. Goto, H. Jane Dyson et al. · Journal of Molecular Biology · 2005 · 171 citations

, , +16

The Transcriptional Activator GCN4 Contains Multiple Activation Domains That Are Critically Dependent on Hydrophobic Amino Acids

Connie M. Drysdale, Encarnación Dueñas, Belinda M. Jackson et al. · Molecular and Cellular Biology · 1995 · 160 citations · Full text

, , +17