Concepedia

Discovery of 1-benzoyl-3-cyanopyrrolo[1,2-a]quinolines as a new series of apoptosis inducers using a cell- and caspase-based high-throughput screening assay. Part 1: Structure–activity relationships of the 1- and 3-positions

William Kemnitzer, Jared Kuemmerle, Songchun Jiang, Han‐Zhong Zhang, Nilantha Sirisoma, Shailaja Kasibhatla, Candace Crogan‐Grundy, Ben Tseng, John Drewe, Sui Xiong Cai

Bioorganic & Medicinal Chemistry Letters · 2008 · 82 citations · 23 references

DOI

Concepts

References

23

The New Era in Cancer Research

Harold Varmus · Science · 2006 · 306 citations

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Antivascular and antitumor evaluation of 2-amino-4-(3-bromo-4,5-dimethoxy-phenyl)-3-cyano-4<i>H</i>-chromenes, a novel series of anticancer agents

Henriette Gourdeau, Lorraine Leblond, Bettina A. Hamelin et al. · Molecular Cancer Therapeutics · 2004 · 289 citations

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Discovery of 4-Aryl-4<i>H</i>-chromenes as a New Series of Apoptosis Inducers Using a Cell- and Caspase-based High-Throughput Screening Assay. 1. Structure−Activity Relationships of the 4-Aryl Group

William Kemnitzer, John Drewe, Songchun Jiang et al. · Journal of Medicinal Chemistry · 2004 · 279 citations

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Discovery and Structure−Activity Relationship of 3-Aryl-5-aryl-1,2,4-oxadiazoles as a New Series of Apoptosis Inducers and Potential Anticancer Agents

Han‐Zhong Zhang, Shailaja Kasibhatla, Jared Kuemmerle et al. · Journal of Medicinal Chemistry · 2005 · 237 citations · Full text

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Discovery, characterization and SAR of gambogic acid as a potent apoptosis inducer by a HTS assay

Han‐Zhong Zhang, Shailaja Kasibhatla, Yan Wang et al. · Bioorganic & Medicinal Chemistry · 2003 · 235 citations

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