Concepedia

Structural basis of the selectivity of the β2-adrenergic receptor for fluorinated catecholamines

Chaya Pooput, Erica Rosemond, Joel Karpiak, Francesca Deflorian, Santiago Vilar, Stefano Costanzi, Jürgen Wess, Kenneth L. Kirk

Bioorganic & Medicinal Chemistry · 2009 · 15 citations · 20 references

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References

20

High-Resolution Crystal Structure of an Engineered Human β <sub>2</sub> -Adrenergic G Protein–Coupled Receptor

Vadim Cherezov, Daniel M. Rosenbaum, Michael A. Hanson et al. · Science · 2007 · 3.3K citations · Full text

, , +17

A STUDY OF THE ADRENOTROPIC RECEPTORS

Raymond P. Ahlquist · American Journal of Physiology-Legacy Content · 1948 · 2.9K citations

, , +8

GPCR Engineering Yields High-Resolution Structural Insights into β <sub>2</sub> -Adrenergic Receptor Function

Daniel M. Rosenbaum, Vadim Cherezov, Michael A. Hanson et al. · Science · 2007 · 1.3K citations

, , +17

Coupling ligand structure to specific conformational switches in the β2-adrenoceptor

Xiao-Jie Yao, Charles Parnot, Xavier Deupí et al. · Nature Chemical Biology · 2006 · 345 citations

, , +14

Sequential Binding of Agonists to the β2 Adrenoceptor

Gayathri Swaminath, Yang K. Xiang, Tae Weon Lee et al. · Journal of Biological Chemistry · 2003 · 331 citations · Full text

, , +17