Concepedia

Identification and SAR of potent and selective non-peptide obeline somatostatin sst1 receptor antagonists

Thomas Troxler, Daniël Hoyer, Daniel Langenegger, Peter Neumann, Paul Pfäffli, Philippe Schoeffter, Dieter Sorg, Robert Swoboda, Konstanze Hurth

Bioorganic & Medicinal Chemistry Letters · 2007 · 10 citations · 28 references

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References

28

Hypothalamic Polypeptide That Inhibits the Secretion of Immunoreactive Pituitary Growth Hormone

Paul Brazeau, Wylie Vale, Roger Burgus et al. · Science · 1973 · 3.5K citations

, , +16

Classification and nomenclature of somatostatin receptors

Daniël Hoyer, G I Bell, Michael Berelowitz et al. · Trends in Pharmacological Sciences · 1995 · 572 citations · Full text

, , +15

Rapid Identification of Subtype-Selective Agonists of the Somatostatin Receptor Through Combinatorial Chemistry

Susan P. Rohrer, Elizabeth T. Birzin, Ralph T. Mosley et al. · Science · 1998 · 461 citations

, , +17

De novo design and synthesis of somatostatin non-peptide peptidomimetics utilizing .beta.-D-glucose as a novel scaffolding

Ralph Hirschmann, K. C. Nicolaou, Sherrie Pietranico et al. · Journal of the American Chemical Society · 1993 · 272 citations

, , +9

Somatostatin regulates dopamine release in rat striatal slices and cat caudate nuclei

MF Chesselet, T Reisine · Journal of Neuroscience · 1983 · 203 citations · Full text

, , +17