Discovery of 2-chloro-N-((4,4-difluoro-1-hydroxycyclohexyl)methyl)-5-(5-fluoropyrimidin-2-yl)benzamide as a potent and CNS penetrable P2X7 receptor antagonist

Xiangyang Chen, Betsy S. Pierce, Win Naing, Margaret L. Grapperhaus, Dennis P. Phillion

Bioorganic & Medicinal Chemistry Letters · 2010 · 38 citations · 11 references

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