Concepedia

Conformationally-flexible benzamide analogues as dopamine D3 and σ2 receptor ligands

Robert H. Mach, Yun‐Sheng Huang, Rebekah A. Freeman, Li Wu, Suwanna Vangveravong, Robert R. Luedtke

Bioorganic & Medicinal Chemistry Letters · 2003 · 93 citations · 14 references

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14

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Distribution of Dopamine D3 Receptor Expressing Neurons in the Human Forebrain Comparison with D2 Receptor Expressing Neurons

Eugenia V. Gurevich · Neuropsychopharmacology · 1999 · 436 citations

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Mesolimbic Dopamine D3 Receptors and Use of Antipsychotics in Patients With Schizophrenia

Eugenia V. Gurevich · Archives of General Psychiatry · 1997 · 249 citations

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Sigma-2 receptors as a biomarker of proliferation in solid tumours

Kenneth T. Wheeler, L-M Wang, C. Anne Wallen et al. · British Journal of Cancer · 2000 · 231 citations · Full text

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Interactive SAR Studies:  Rational Discovery of Super-Potent and Highly Selective Dopamine D3 Receptor Antagonists and Partial Agonists

Laura Bettinetti, Karin Schlotter, Harald Hübner et al. · Journal of Medicinal Chemistry · 2002 · 194 citations · Full text

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