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2-Aryl tryptamines: selective high-affinity antagonists for the h5-HT2A receptor

Graeme I. Stevenson, Adrian L. Smith, Stephen J. Lewis, Stephen G. Michie, Joseph G. Neduvelil, Smita S. Patel, Rosemarie Marwood, Shil Patel, José L. Castro

Bioorganic & Medicinal Chemistry Letters · 2000 · 84 citations · 7 references

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References

7

2-Substituted Tryptamines:  Agents with Selectivity for 5-HT<sub>6</sub>Serotonin Receptors

Richard A. Glennon, Mase Lee, Jagadeesh B. Rangisetty et al. · Journal of Medicinal Chemistry · 2000 · 149 citations · Full text

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Signal transduction differences between 5-hydroxytryptamine type 2A and type 2C receptor systems.

Kelly A. Berg, William P. Clarke, Cynthia Sailstad et al. · Molecular Pharmacology · 1994 · 132 citations

, , +17

Rapid purification of small molecule libraries by ion exchange chromatography

Miles G. Siegel, Patric J. Hahn, Bruce A. Dressman et al. · Tetrahedron Letters · 1997 · 127 citations

, , +16

Relative affinities of drugs acting at cholinoceptors in displacing agonist and antagonist radioligands: the NMS/Oxo‐M ratio as an index of efficacy at cortical muscarinic receptors

Stephen B. Freedman, Elizabeth A. Harley, Leslie L. Iversen · British Journal of Pharmacology · 1988 · 109 citations · Full text

, , +17

Solid-phase synthesis of 2,3-disubstituted indoles: discovery of a novel, high-affinity, selective h5-HT2A antagonist

Adrian L. Smith, Graeme I. Stevenson, Stephen J. Lewis et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 51 citations · Full text

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