New 1,2,3-triazolo[1,5-a]quinoxalines: synthesis and binding to benzodiazepine and adenosine receptors. II

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

Life Sciences, Biochemistry, Chemical Kinetics +14

Development of a comprehensive pharmacophore model for the benzodiazepine receptor.

W Zhang, Konrad F. Koehler, Puhong Zhang et al. · PubMed · 1995 · 93 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Current Developments of A2a Adenosine Receptor Antagonists

Pier Giovanni Baraldi, B. Cacciar, Giampiero Spalluto et al. · Current Medicinal Chemistry · 1995 · 57 citations

Medicine, Medicinal Chemistry, Pharmacology +8

[³H]Muscimol Binding Site on Purified Benzodiazepine Receptor

Claudia Martini, T. Rigacci, Antonio Lucacchini · Journal of Neurochemistry · 1983 · 57 citations

Medicine, Neuroscience, Pharmacology +13

Potential antileukemic and immunosuppressive drugs. 3. Effects of homocyclic ring substitution on the in vitro drug activity of 4-nitrobenzo-2,1,3-oxadiazoles (4-nitrobenzofurazans) and their N-oxides (4-nitrobenzofuroxans)

P. B. Ghosh, B. Ternai, M. W. Whitehouse · Journal of Medicinal Chemistry · 1972 · 55 citations

Pharmacy, Medicinal Chemistry, Pharmacology +8