Concepedia

SB-236057, a selective 5-HT1B receptor inverse agonist, blocks the 5-HT human terminal autoreceptor

Derek N. Middlemiss, Manfred Göthert, Eberhard Schlicker, Claire M. Scott, Julie V. Selkirk, Jeanette Watson, Laramie M. Gaster, Paul Wyman, Graham J. Riley, Gary Price

European Journal of Pharmacology · 1999 · 39 citations · 14 references

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14

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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SB-216641 and BRL-15572 – compounds to pharmacologically discriminate h5-HT1B and h5-HT1D receptors

Gary Price, Melanie J. Burton, L. J. Collin et al. · Naunyn-Schmiedeberg s Archives of Pharmacology · 1997 · 167 citations · Full text

, , +14

Effect of a selective 5‐HT reuptake inhibitor in combination with 5‐HT<sub>1A</sub> and 5‐HT<sub>1B</sub> receptor antagonists on extracellular 5‐HT in rat frontal cortex <i>in vivo</i>

Trevor Sharp, Valerie Umbers, Sarah E. Gartside · British Journal of Pharmacology · 1997 · 136 citations · Full text

, , +17

SB‐224289–a novel selective (human) 5‐HT<sub>1B</sub> receptor antagonist with negative intrinsic activity

Julie V. Selkirk, Claire M. Scott, M Ho et al. · British Journal of Pharmacology · 1998 · 125 citations · Full text

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Stimulation of 5-HT1B receptors causes hypothermia in the guinea pig

Jim J. Hagan, Paula D. Slade, Laramie M. Gaster et al. · European Journal of Pharmacology · 1997 · 96 citations

, , +9