Design and SAR of macrocyclic Hsp90 inhibitors with increased metabolic stability and potent cell-proliferation activity - Concepedia

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Design and SAR of macrocyclic Hsp90 inhibitors with increased metabolic stability and potent cell-proliferation activity

DOI Full Paper Access

24

Citations

13

References

2011

Year

Christoph W. Zapf, Jonathan D. Bloom, Jamie L. McBean, Russell G. Dushin, Thomas Nittoli, Charles L. Ingalls, Alan G. Sutherland, John P. Sonye, Clark N. Eid, Jennifer M. Golas,

Bioorganic & Medicinal Chemistry Letters

Macrocyclic Hsp90 InhibitorsDrug TargetMedicineRational Drug DesignPotent Cell-proliferation ActivityIncreased Metabolic StabilityAnti-cancer AgentDrug DevelopmentPharmacologyRadiation OncologyTumor MicroenvironmentDrug Discovery

References

	Year	Citations

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