Concepedia

The effect of 17-N substituents on the activity of the opioid κ receptor in nalfurafine derivatives

Toru Nemoto, Naoshi Yamamoto, Naohisa Wada, Yukimasa Harada, Miyuki Tomatsu, Marina Ishihara, Shigeto Hirayama, Takashi Iwai, H. Fujii, Hiroshi Nagase

Bioorganic & Medicinal Chemistry Letters · 2012 · 21 citations · 18 references

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References

18

U-50,488: a selective and structurally novel non-Mu (kappa) opioid agonist.

Philip F. VonVoigtlander, Robert A. Lahti, James H. Ludens · Journal of Pharmacology and Experimental Therapeutics · 1983 · 816 citations

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A mild, general method for conversion of esters to amides

Anwer Basha, Michael F. Lipton, Steven M. Weinreb · Tetrahedron Letters · 1977 · 560 citations

, , +3

Synthetic Analgesics: Stereochemical Considerations

A H Beckett, A. F. Casy · Journal of Pharmacy and Pharmacology · 1954 · 332 citations

, , +17

Properties of a selective kappa agonist, U-50,488H

Robert A. Lahti, Philip F. VonVoigtlander, Craig L. Barsuhn · Life Sciences · 1982 · 198 citations

, , +8

Discovery of a Structurally Novel Opioid .KAPPA.-Agonist Derived from 4,5-Epoxymorphinan.

Hiroshi Nagase, Jun Hayakawa, Kuniaki Kawamura et al. · Chemical and Pharmaceutical Bulletin · 1998 · 188 citations · Full text

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