Concepedia

Hydroxylated 2,3-diarylindenes: Synthesis, estrogen receptor binding affinity, and binding orientation considerations

Gregory M. Anstead, Chad S. Peterson, John A. Katzenellenbogen

Journal of Steroid Biochemistry · 1989 · 20 citations · 24 references

DOI

Concepts

References

24

Rapid chromatographic technique for preparative separations with moderate resolution

W. Clark Still, Michaël Kahn, Abhijit Mitra · The Journal of Organic Chemistry · 1978 · 5.8K citations

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Hydrogen bonding and biological specificity analysed by protein engineering

Alan R. Fersht, Jianping Shi, J.W. Knill-Jones et al. · Nature · 1985 · 1.1K citations

, , +16

Antiestrogens. 2. Structure-activity studies in a series of 3-aroyl-2-arylbenzo[b]thiophene derivatives leading to [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl]-[4-[2-(1-piperidinyl)ethoxy]phenyl]methanone hydrochloride (LY 156758), a remarkably effective estrogen antagonist with only minimal intrinsic estrogenicity

Charles D. Jones, Mary G. Jevnikar, Andrew Pike et al. · Journal of Medicinal Chemistry · 1984 · 285 citations

, , +7

Relation Between Estrogen Inhibitory Activity and Binding to Cytosol of Rabbit and Human Uterus

Stanley G. Korenman · Endocrinology · 1970 · 243 citations

, , +12

Photoaffinity labels for estrogen binding proteins of rat uterus

John A. Katzenellenbogen, Howard J. Johnson, Harvey N. Myers · Biochemistry · 1973 · 219 citations

, , +11