Concepedia

N-[4-(Methylsulfonylamino)benzyl]thiourea analogues as vanilloid receptor antagonists: analysis of structure–activity relationships for the ‘C-Region’

Jeewoo Lee, Sang-Uk Kang, Ju‐Ok Lim, Hyun‐Kyung Choi, Mi-Kyung Jin, Attila Tóth, Larry V. Pearce, Richard Tran, Yun Wang, Tamás Szabó,

Bioorganic & Medicinal Chemistry · 2003 · 34 citations · 28 references

DOI

Concepts

References

28

The capsaicin receptor: a heat-activated ion channel in the pain pathway

Michael J. Caterina, Mark Schumacher, Makoto Tominaga et al. · Nature · 1997 · 9.1K citations

, , +16

The Cloned Capsaicin Receptor Integrates Multiple Pain-Producing Stimuli

Makoto Tominaga, Michael J. Caterina, Annika B. Malmberg et al. · Neuron · 1998 · 3.1K citations · Full text

, , +14

Vanilloid receptors on sensory nerves mediate the vasodilator action of anandamide

Peter M. Zygmunt, Jesper Petersson, David A. Andersson et al. · Nature · 1999 · 2.1K citations

, , +10

Direct activation of capsaicin receptors by products of lipoxygenases: Endogenous capsaicin-like substances

Sun Wook Hwang, Hawon Cho, Jiyeon Kwak et al. · Proceedings of the National Academy of Sciences · 2000 · 1K citations

, , +17

Capsazepine: a competitive antagonist of the sensory neurone excitant capsaicin

Stuart Bevan, Sandeep S Hothi, Glyn A. Hughes et al. · British Journal of Pharmacology · 1992 · 584 citations · Full text

, , +16