Publication | Open Access
Computationally motivated synthesis and enzyme kinetic evaluation of N-(β-<scp>d</scp>-glucopyranosyl)-1,2,4-triazolecarboxamides as glycogen phosphorylase inhibitors
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Citations
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References
2014
Year
GlycobiologyEnzymatic ModificationPharmaceutical ChemistryEnzyme Kinetic EvaluationMolecular PharmacologyMedicinal ChemistryInhibitory ActivityGlycosylationBiochemistryMechanism Of ActionGlycogen Phosphorylase BDrug DevelopmentPharmacologyMolecular ModelingNatural SciencesRational Drug DesignGlycogen Phosphorylase InhibitorsMedicineDrug Discovery
<italic>N</italic>-(β-<sc>d</sc>-Glucopyranosyl)-1,2,4-triazolecarboxamides discovered as low μM inhibitors of glycogen phosphorylase b.
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