N-Cbz sulfilimines as valuable intramolecular nucleophiles for the stereoselective synthesis of (−)-deoxocassine and (+)-desoxoprosophylline

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Naoki Asano, Robert J. Nash, Russell J. Molyneux et al. · Tetrahedron Asymmetry · 2000 · 1K citations

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Effect of the acidic component on the Mitsunobu inversion of a sterically hindered alcohol

Jeffrey A. Dodge, John I. Trujillo, Misti Presnell · The Journal of Organic Chemistry · 1994 · 159 citations

Natural Sciences, Chemistry, Medicinal Chemistry +6

Construction of Hydroxylated Alkaloids (.+-.)-Mannonolactam, (.+-.)-Deoxymannojirimycin, and (.+-.)-Prosopinine through Aza-Annulation

Gregory R. Cook, Lars G. Beholz, John R. Stille · The Journal of Organic Chemistry · 1994 · 118 citations

Natural Sciences, Chemistry, Medicinal Chemistry +9

Rhodium-Catalyzed Cyclohydrocarbonylation:  Application to the Synthesis of (+)-Prosopinine and (−)-Deoxoprosophylline

Iwao Ojima, Ephraim S. Vidal · The Journal of Organic Chemistry · 1998 · 94 citations

Natural Sciences, Chemistry, Medicinal Chemistry +9

A Novel Regio- and Stereoselective Synthesis of Sulfamidates from 1,2-Diols Using Burgess and Related Reagents: A Facile Entry into β-Amino Alcohols We thank Professor K. Barry Sharpless for the gracious donation of several of the starting diol substrates. We also thank Drs. D. H. Huang, G. Suizdak, and R. Chadja for NMR spectroscopic, mass spectrometric, and X-ray crystallographic assistance, respectively. Financial support for this work was provided by The Skaggs Institute for Chemical Biology, predoctoral fellowships from the National Science Foundation and Pfizer (S.A.S.), a postdoctoral fellowship from The Skaggs Institute for Chemical Biology (X.H.), and grants from American Biosciences, Amgen, Array Biopharma, Boehringer-Ingelheim, Glaxo, Hoffman-LaRoche, DuPont, Merck, Novartis, Pfizer, and Schering Plough.

K. C. Nicolaou, Xianhai Huang, Scott A. Snyder et al. · Angewandte Chemie International Edition · 2002 · 86 citations

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