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Synthesis of new glycosyl biuret and urea derivatives as potential glycoenzyme inhibitors

Nóra Felföldi, Marietta Tóth, Evangelia D. Chrysina, Maria-Despoina Charavgi, K.-M. Alexacou, László Somsák

Carbohydrate Research · 2009 · 17 citations · 17 references

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17

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Assay of inorganic phosphate in the mild pH range, suitable for measurement of glycogen phosphorylase activity

Shuichi Saheki, Akira Takeda, Takashi Shimazu · Analytical Biochemistry · 1985 · 217 citations

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Carbohydrate-based drug discovery.

Chi-Huey Wong · 2003 · 202 citations

Binding of <i>N</i>‐acetyl‐<i>N</i> ′‐β‐<scp>d</scp>‐glucopyranosyl urea and <i>N</i>‐benzoyl‐<i>N</i> ′‐β‐<scp>d</scp>‐glucopyranosyl urea to glycogen phosphorylase <i>b</i>

Nikos G. Oikonomakos, Magda Kosmopoulou, S.E. Zographos et al. · European Journal of Biochemistry · 2002 · 70 citations · Full text

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A new, scalable preparation of a glucopyranosylidene-spiro-thiohydantoin: one of the best inhibitors of glycogen phosphorylases

László Somsák, Véronika Nagy · Tetrahedron Asymmetry · 2000 · 61 citations · Full text

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