Concepedia

Isoxazole analogues bind the System xc- transporter: Structure–activity relationship and pharmacophore model

Sarjubhai A. Patel, Trideep Rajale, Erin M. O’Brien, David J. Burkhart, Jared K. Nelson, Brendan Twamley, Alex Blumenfeld, Monika I. Szabon-Watola, John M. Gerdes, Richard J. Bridges,

Bioorganic & Medicinal Chemistry · 2009 · 30 citations · 39 references

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References

39

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Neuroadaptations in cystine-glutamate exchange underlie cocaine relapse

David L. Baker, Krista McFarland, RUSSELL W. LAKE et al. · Nature Neuroscience · 2003 · 743 citations

, , +12

The Origin and Neuronal Function of<i>In Vivo</i>Nonsynaptic Glutamate

David L. Baker, Zheng‐Xiong Xi, Hui Shen et al. · Journal of Neuroscience · 2002 · 583 citations · Full text

, , +17

Exchange of cystine and glutamate across plasma membrane of human fibroblasts.

Shiro Bannai · Journal of Biological Chemistry · 1986 · 537 citations · Full text

, , +6

Calcium‐Dependent and‐Independent Release of Glutamate from Synaptosomes Monitored by Continuous Fluorometry

David G. Nicholls, Talvinder S. Sihra, José Sánchez‐Prieto · Journal of Neurochemistry · 1987 · 463 citations

, , +17