Concepedia

Improved synthesis of (S)-7-amino-5H,7H-dibenzo[b,d]azepin-6-one, a building block for γ-secretase inhibitors

Fabienne Hoffmann-Emery, Roland Jakob‐Roetne, Alexander Flohr, Fritz Bliss, Reinhard Reents

Tetrahedron Letters · 2009 · 15 citations · 4 references

DOI

Concepts

References

4

Application of the Palladium-Catalyzed Borylation/Suzuki Coupling (BSC) Reaction to the Synthesis of Biologically Active Biaryl Lactams

Olivier Baudoin, Michèle Césario, Daniel Guénard et al. · The Journal of Organic Chemistry · 2002 · 231 citations

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A multigram chemical synthesis of the γ-secretase inhibitor LY411575 and its diastereoisomers

Abdul H. Fauq, Katherine Simpson, Ghulam M. Maharvi et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 74 citations · Full text

, , +12

Highly efficient synthesis of medium-sized lactams via intramolecular Staudinger–aza-Wittig reaction of ω-azido pentafluorophenyl ester: synthesis and biological evaluation of LY411575 analogues

Haruhiko Fuwa, Yumiko Okamura, Yuichi Morohashi et al. · Tetrahedron Letters · 2004 · 45 citations

, , +10

Synthesis of Dimethylapoerysopine and an Approach to the Total Synthesis of the Unrearranged Erythrina Bases

K. Wiesner, Z. Valenta, A. J. Manson et al. · Journal of the American Chemical Society · 1955 · 39 citations

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