Concepedia

Interaction of the Novel Adenosine Uptake Inhibitor 3-[1-(6,7-Diethoxy-2-morpholinoquinazolin-4-yl)piperidin-4-yl]-1,6-dimethyl-2,4(1 H,3 H)-quinazolinedione Hydrochloride (KF24345) with the es and ei Subtypes of Equilibrative Nucleoside Transporters

James R. Hammond, Richard G. E. Archer

Journal of Pharmacology and Experimental Therapeutics · 2004 · 20 citations · 28 references

DOI

Concepts

References

28

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

The preparation and chemical characteristics of hemoglobin-free ghosts of human erythrocytes

James T. Dodge, Carolyn D. Mitchell, Donald J. Hanahan · Archives of Biochemistry and Biophysics · 1963 · 4.4K citations

, , +8

Cloning of a human nucleoside transporter implicated in the Cellular uptake of adenosine and chemotherapeutic drugs

Mark Griffiths, Nick Beaumont, Sylvia Y.M. Yao et al. · Nature Medicine · 1997 · 426 citations

, , +13

The control of the metabolism and the hormonal role of adenosine.

J R Arch, Eric A. Newsholme · PubMed · 1978 · 415 citations

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Kinetic and Pharmacological Properties of Cloned Human Equilibrative Nucleoside Transporters, ENT1 and ENT2, Stably Expressed in Nucleoside Transporter-deficient PK15 Cells

Jeffrey L. Ward, Azeem Sherali, Zhi-Ping Mo et al. · Journal of Biological Chemistry · 2000 · 315 citations · Full text

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