Concepedia

Synthesis and in vivo evaluation of bicyclic gababutins

David C. Blakemore, Justin S. Bryans, Pauline Carnell, Christopher L. Carr, N. Chessum, Mark J. Field, Natasha Kinsella, Simon A. Osborne, Andrew N. Warren, Sophie C. Williams

Bioorganic & Medicinal Chemistry Letters · 2009 · 37 citations · 7 references

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7

The Novel Anticonvulsant Drug, Gabapentin (Neurontin), Binds to the α2δ Subunit of a Calcium Channel

N S Gee, Jason P. Brown, Visaka U.K. Dissanayake et al. · Journal of Biological Chemistry · 1996 · 1.2K citations · Full text

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Gabapentin in postherpetic neuralgia: a randomised, double blind, placebo controlled study

Andrew S.C. Rice, S. Maton · Pain · 2001 · 596 citations

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Structure−Activity Relationships of Pregabalin and Analogues That Target the α<sub>2</sub>-δ Protein

Thomas R. Belliotti, Thomas Capiris, I. Victor Ekhato et al. · Journal of Medicinal Chemistry · 2005 · 210 citations

, , +17

Mechanism of Action of α<sub>2</sub>δ Ligands: Voltage Sensitive Calcium Channel (VSCC) Modulators

Stephen M. Stahl · The Journal of Clinical Psychiatry · 2004 · 64 citations

, , +17

Biocatalytic preparation of bicyclo[3.2.0]heptane derivatives

Norbert Klempier, Paul Geymayer, Peter Stadler et al. · Tetrahedron Asymmetry · 1990 · 27 citations

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