Concepedia
Bioorganic & Medicinal Chemistry · 2012 · 58 citations · 23 references
Open access
Protein ChemistryMolecular PharmacologyBiochemistryMedicineNatural SciencesBioanalysisChemical BiologyPharmacologyInhibitor BindingCarbonyl Metabolism
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Carbonic anhydrase inhibitors
Claudiu T. Supuran, Andrea Scozzafava, Angela Casini · Medicinal Research Reviews · 2002 · 1.4K citations
Hypoxia-Inducible Carbonic Anhydrase IX and XII Promote Tumor Cell Growth by Counteracting Acidosis through the Regulation of the Intracellular pH
Johanna Chiche, Karine Ilc, Julie Laferrière et al. · Cancer Research · 2008 · 727 citations
Thermodynamic Stability of Carbonic Anhydrase: Measurements of Binding Affinity and Stoichiometry Using ThermoFluor
Daumantas Matulis, James K. Kranz, F. Raymond Salemme et al. · Biochemistry · 2005 · 486 citations
Engineering, Protein Assembly, Binding Affinity +22
Deciphering the Mechanism of Carbonic Anhydrase Inhibition with Coumarins and Thiocoumarins
Alfonso Maresca, Claudia Temperini, Lionel Pochet et al. · Journal of Medicinal Chemistry · 2009 · 395 citations · Full text
Evaluation of linked protonation effects in protein binding reactions using isothermal titration calorimetry
Brian M. Baker, Kenneth P. Murphy · Biophysical Journal · 1996 · 335 citations · Full text
Protein Chemistry, Engineering, Biochemistry +11