First synthesis of P-aryl-phosphinosugars, organophosphorus analogues of C-arylglycosides

New hybrid transition state analog inhibitors of HIV protease with peripheric C2-symmetry

Bernd Stowasser, Karl‐Heinz Budt, Jianqi Li et al. · Tetrahedron Letters · 1992 · 407 citations

Life Sciences, Medicinal Chemistry, Molecular Biology +13

The Most Potent Organophosphorus Inhibitors of Leucine Aminopeptidase. Structure-Based Design, Chemistry, and Activity

Jolanta Grembecka, Artur Mucha, Tomasz Cierpicki et al. · Journal of Medicinal Chemistry · 2003 · 221 citations · Full text

Life Sciences, Biochemistry, Pharmacology +12

Inhibition of aminopeptidases by aminophosphonates

Barbara Lejczak, Paweł Kafarski, Jan Zygmunt · Biochemistry · 1989 · 133 citations

Life Sciences, Biochemistry, Pharmacology +8

Inhibition of human immunodeficiency virus-1 protease by a C2-symmetric phosphinate. Synthesis and crystallographic analysis

Sherin S. Abdel‐Meguid, Baoguang Zhao, Krishna H. M. Murthy et al. · Biochemistry · 1993 · 77 citations

Life Sciences, Biochemistry, Molecular Biology +16

Cyclic Phosphonate Analogs of Hexopyranoses

James W. Darrow, Dale G. Drueckhammer · The Journal of Organic Chemistry · 1994 · 73 citations

Natural Sciences, Chemistry, Analytical Chemistry +4