Concepedia

Design, synthesis, and structure–activity relationship of novel opioid κ-agonists

Koji Kawai, Jun Hayakawa, Toru Miyamoto, Yoshifumi Imamura, Shinichi Yamane, Hisanori Wakita, H. Fujii, Kuniaki Kawamura, Hirotoshi Matsuura, Naoki Izumimoto,

Bioorganic & Medicinal Chemistry · 2008 · 75 citations · 26 references

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References

26

Application of the message-address concept in the design of highly potent and selective non-peptide .delta. opioid receptor antagonists

P. S. Portoghese, Marjia Sultana, Hiroshi Nagase et al. · Journal of Medicinal Chemistry · 1988 · 305 citations

, , +15

Antipruritic activity of the κ-opioid receptor agonist, TRK-820

Yuko Togashi, Hideo Umeuchi, Kiyoshi Okano et al. · European Journal of Pharmacology · 2002 · 207 citations

, , +13

Discovery of a Structurally Novel Opioid .KAPPA.-Agonist Derived from 4,5-Epoxymorphinan.

Hiroshi Nagase, Jun Hayakawa, Kuniaki Kawamura et al. · Chemical and Pharmaceutical Bulletin · 1998 · 188 citations · Full text

, , +17

Blockade of morphine reward through the activation of κ-opioid receptors in mice

Masahiko Funada, Tsutomu Suzuki, Minoru Narita et al. · Neuropharmacology · 1993 · 167 citations

, , +14

Benzeneacetamide amines: structurally novel non-m.mu. opioids

Jacob Szmuszkovicz, P. F. VON VOIGTLANDER · Journal of Medicinal Chemistry · 1982 · 155 citations

, , +6