Concepedia

Synthesis and evaluation of cis-hexahydropyrrolo[3,2-b]pyrrol-3-one peptidomimetic inhibitors of CAC1 cysteinyl proteinases

Martin Quibell, Alex Benn, Nick Flinn, Tracy Monk, Manoj K. Ramjee, Peter C. Ray, Yikang Wang, John P. Watts

Bioorganic & Medicinal Chemistry · 2004 · 12 citations · 37 references

DOI

Concepts

References

37

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

Christopher A. Lipinski, Franco Lombardo, Beryl W. Dominy et al. · Advanced Drug Delivery Reviews · 1997 · 11.2K citations

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Molecular Properties That Influence the Oral Bioavailability of Drug Candidates

Daniel F. Veber, Stephen R. Johnson, Hung‐Yuan Cheng et al. · Journal of Medicinal Chemistry · 2002 · 8.1K citations

, , +15

The Handbook of proteolytic enzymes

A. John Barrett, Neil D. Rawlings, J. Frederick Woessner · 1998 · 1.1K citations

, , +12

New coupling reagents in peptide chemistry

Reinhard Knorr, Arnold Trzeciak, Willi Bannwarth et al. · Tetrahedron Letters · 1989 · 986 citations

, , +8

Solid phase peptide synthesis; a practical approach

Comparative Biochemistry and Physiology Part A Physiology · 1991 · 762 citations

, , +5