Concepedia

Design, synthesis, and biological evaluation of 4-arylmethyl-1-phenylpyrazole and 4-aryloxy-1-phenylpyrazole derivatives as novel androgen receptor antagonists

Satoshi Yamamoto, Naoki Tomita, Yuri Suzuki, Tomohiko Suzaki, Tomohiro Kaku, Takahito Hara, Masuo Yamaoka, Naoyuki Kanzaki, Atsushi Hasuoka, Atsuo Baba,

Bioorganic & Medicinal Chemistry · 2012 · 28 citations · 28 references

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28

Cancer Statistics, 2008

Ahmedin Jemal, Rebecca L. Siegel, Elizabeth Ward et al. · CA A Cancer Journal for Clinicians · 2008 · 10.2K citations · Full text

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Docetaxel plus Prednisone or Mitoxantrone plus Prednisone for Advanced Prostate Cancer

Ian F. Tannock, Ronald de Wit, William R. Berry et al. · New England Journal of Medicine · 2004 · 5.7K citations

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Development of a Second-Generation Antiandrogen for Treatment of Advanced Prostate Cancer

Chris Tran, Samedy Ouk, Nicola J. Clegg et al. · Science · 2009 · 2.3K citations · Full text

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Molecular determinants of resistance to antiandrogen therapy

Charlie D. Chen, Derek S. Welsbie, Chris Tran et al. · Nature Medicine · 2003 · 2.3K citations

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A Biological Profile of a Nonsteroidal Antiandrogen, SCH 13521 (4'–Nitro–3'–Trifluoromethylisobutyranilide)1

R. Neri, KATHERYN FLORANCE, Patricia Koziol et al. · Endocrinology · 1972 · 327 citations

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