Bioorganic & Medicinal Chemistry · 2013 · 33 citations · 25 references
PharmacyMedicinal ChemistryPharmacologyDrug DiscoveryOrganic ChemistryStructure-activity RelationshipsEnzyme InhibitionGabaergic NeurochemistryGabaergic PharmacologyGabaergic SignalingHeterocyclic ChemistryStructure-activity Relationship AnalysisGaba AntagonistsGaba Receptor AntagonismGaba Uptake InhibitionGaba-b Receptor PharmacologyGabaergic Drug DiscoveryGabaergic Neurotransmission ModulationMedicinal Chemistry Applications
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Cloning and Expression of a Rat Brain GABA Transporter
John Guastella, Nathan Nelson, Hannah Nelson et al. · Science · 1990 · 881 citations
Qing‐Rong Liu, Beatriz López‐Corcuera, Sreekala Mandiyan et al. · Journal of Biological Chemistry · 1993 · 419 citations · Full text