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Synthesis of Imidazopyridines and Purines as Potent Inhibitors of Leukotriene A4 Hydrolase

Thomas D. Penning, Nizal S. Chandrakumar, B.N. Desai, Stevan W. Djurić, Alan F. Gasiecki, James W. Malecha, Julie M. Miyashiro, Mark A. Russell, Leslie J. Askonas, James K. Gierse,

Bioorganic & Medicinal Chemistry Letters · 2003 · 28 citations · 9 references

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9

An improved synthesis of homoproline and derivatives

Robert T. Shuman, Paul L. Ornstein, Jonathan W. Paschal et al. · The Journal of Organic Chemistry · 1990 · 85 citations

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Structure−Activity Relationship Studies on 1-[2-(4-Phenylphenoxy)ethyl]pyrrolidine (SC-22716), a Potent Inhibitor of Leukotriene A<sub>4</sub> (LTA<sub>4</sub>) Hydrolase

Thomas D. Penning, Nizal S. Chandrakumar, Barbara B. Chen et al. · Journal of Medicinal Chemistry · 2000 · 68 citations · Full text

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Pharmacological Characterization of SC-57461A (3-[Methyl[3-[4-(phenylmethyl)phenoxy]propyl]amino]propanoic Acid HCl), a Potent and Selective Inhibitor of Leukotriene A4Hydrolase I: In Vitro Studies

Leslie J. Askonas, James F. Kachur, Doreen Villani-Price et al. · Journal of Pharmacology and Experimental Therapeutics · 2002 · 47 citations

, , +13

Synthesis of Potent Leukotriene A<sub>4</sub> Hydrolase Inhibitors. Identification of 3-[Methyl[3-[4-(phenylmethyl)phenoxy]propyl]amino]propanoic Acid

Thomas D. Penning, Mark A. Russell, Barbara B. Chen et al. · Journal of Medicinal Chemistry · 2002 · 39 citations · Full text

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Improved Procedures for Preparation of 2-Pyridones and 2-Hydroxymethylpyridines from Pyridine N-Oxides

Katsuhiro Konno, Kimiko Hashimoto, Hatuhisa Shirahama et al. · Heterocycles · 1986 · 37 citations · Full text

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