Medicinal Chemistry Research · 2012 · 24 citations · 31 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryPharmacophore ModelingLigand BindingMechanisms Of Drug ActionPharmacophore MappingPotency OptimizationQuantitative Structure-activity RelationshipsStructure-based Pharmacophore ModelingKappa Opioid Receptor PharmacologyOpioid AntagonistsOpioid Receptor AgonistsOpioid Receptor BindingReceptor Binding ModelsReceptor-based Pharmacophore Generation
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Principles of QSAR models validation: internal and external
Paola Gramatica · QSAR & Combinatorial Science · 2007 · 2.2K citations · Full text