Concepedia

N-4-Substituted-benzyl-N′-tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activity

Hyeung‐geun Park, JiYeon Choi, Sea‐hoon Choi, Mi-Kyung Park, Jihye Lee, Young‐Ger Suh, Hawon Cho, Uhtaek Oh, Jiyoun Lee, Sang-Uk Kang,

Bioorganic & Medicinal Chemistry Letters · 2004 · 27 citations · 24 references

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References

24

The capsaicin receptor: a heat-activated ion channel in the pain pathway

Michael J. Caterina, Mark Schumacher, Makoto Tominaga et al. · Nature · 1997 · 9.1K citations

, , +16

The Cloned Capsaicin Receptor Integrates Multiple Pain-Producing Stimuli

Makoto Tominaga, Michael J. Caterina, Annika B. Malmberg et al. · Neuron · 1998 · 3.1K citations · Full text

, , +14

Capsaicin-induced ion fluxes in dorsal root ganglion cells in culture

JN Wood, J. Winter, I. F. James et al. · Journal of Neuroscience · 1988 · 566 citations · Full text

, , +17

Iodo-Resiniferatoxin, a New Potent Vanilloid Receptor Antagonist

Philip Wahl, Christian Foged, Søren Tullin et al. · Molecular Pharmacology · 2001 · 253 citations

, , +11

The Discovery of Capsazepine, the First Competitive Antagonist of the Sensory Neuron Excitants Capsaicin and Resiniferatoxin

Christopher Walpole, Stuart Bevan, G. Bovermann et al. · Journal of Medicinal Chemistry · 1994 · 210 citations

, , +16