Concepedia

Functionalized pyrrolidine inhibitors of human type II α-mannosidases as anti-cancer agents: Optimizing the fit to the active site

Hélène Fiaux, D.A. Kuntz, Daniela Hoffman, Robert C. Janzer, Sandrine Gerber‐Lemaire, David R. Rose, Lucienne Juillerat‐Jeanneret

Bioorganic & Medicinal Chemistry · 2008 · 56 citations · 31 references

DOIFull text

Open access

Concepts

References

31

[16] SHELXL: High-resolution refinement

George M. Sheldrick, T. Schneider · Methods in enzymology on CD-ROM/Methods in enzymology · 1997 · 2.5K citations

, , +4

Sugar-mimic glycosidase inhibitors: natural occurrence, biological activity and prospects for therapeutic application

Naoki Asano, Robert J. Nash, Russell J. Molyneux et al. · Tetrahedron Asymmetry · 2000 · 1K citations

, , +17

A Spectroscopic Investigation of Swainsonine: An α-Mannosidase Inhibitor Isolated from <i>Swainsona canescens</i>

SM Colegate, PR Dorling, CR Huxtable · Australian Journal of Chemistry · 1979 · 425 citations

, , +9

Structure of Golgi α‐mannosidase II: a target for inhibition of growth and metastasis of cancer cells

Jean van den Elsen · The EMBO Journal · 2001 · 217 citations · Full text

, , +14

Assignment of the Absolute Configuration of Natural Lentiginosine by Synthesis and Enzymic Assays of Optically Pure (+) and (-)-Enantiomers

Alberto Brandi, Stefano Cicchi, Franca M. Cordero et al. · The Journal of Organic Chemistry · 1995 · 195 citations · Full text

, , +9