Concepedia

Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a

Jean-Philippe Leyris, Thomas Roux, Eric Trinquet, Pascal Verdié, Jean‐Alain Fehrentz, Nadia Oueslati, Stéphanie Douzon, Emmanuel Bourrier, Laurent Lamarque, Didier Gagne,

Analytical Biochemistry · 2010 · 82 citations · 32 references

DOI

Concepts

References

32

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.8K citations

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THE PREPARATION OF 131I-LABELLED HUMAN GROWTH HORMONE OF HIGH SPECIFIC RADIOACTIVITY

FC Greenwood, WM Hunter, J. Glover · Biochemical Journal · 1963 · 10.2K citations · Full text

, , +11

Preparation of Iodine-131 Labelled Human Growth Hormone of High Specific Activity

W. M. Hunter, F. C. Greenwood · Nature · 1962 · 7K citations

, , +8

The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints

Robert Fredriksson, Malin C. Lagerström, Lars‐Gustav Lundin et al. · Molecular Pharmacology · 2003 · 2.9K citations

High Constitutive Signaling of the Ghrelin Receptor—Identification of a Potent Inverse Agonist

Birgitte Holst, Adam I. Cygankiewicz, Tine H. Jensen et al. · Molecular Endocrinology · 2003 · 510 citations