Concepedia

Facile transformation of Biginelli pyrimidin-2(1H)-ones to pyrimidines. In vitro evaluation as inhibitors of Mycobacterium tuberculosis and modulators of cytostatic activity

Kamaljit Singh, Kawaljit Singh, Kawaljit Singh, Baojie Wan, Scott G. Franzblau, Kelly Chibale, Jan Balzarini

European Journal of Medicinal Chemistry · 2011 · 76 citations · 17 references

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References

17

Microplate alamar blue assay versus BACTEC 460 system for high-throughput screening of compounds against Mycobacterium tuberculosis and Mycobacterium avium

L A Collins, Scott G. Franzblau · Antimicrobial Agents and Chemotherapy · 1997 · 1.6K citations · Full text

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100 years of the biginelli dihydropyrimidine synthesis

C. Oliver Kappe · Tetrahedron · 1993 · 1.2K citations

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DNA gyrase, topoisomerase IV, and the 4-quinolones.

Karl Drlica, Xilin Zhao · Microbiology and Molecular Biology Reviews · 1997 · 891 citations

, , +11

PA-824 Kills Nonreplicating <i>Mycobacterium tuberculosis</i> by Intracellular NO Release

Ramandeep Singh, Ujjini H. Manjunatha, Helena I. Boshoff et al. · Science · 2008 · 635 citations · Full text

, , +14

Studies on the Mechanism of Action of Isoniazid and Ethionamide in the Chemotherapy of Tuberculosis

Kai Johnsson, David S. King, Peter G. Schultz · Journal of the American Chemical Society · 1995 · 213 citations · Full text

, , +9