Kawaljit Singh

Facile transformation of Biginelli pyrimidin-2(1H)-ones to pyrimidines. In vitro evaluation as inhibitors of Mycobacterium tuberculosis and modulators of cytostatic activity

Kamaljit Singh, Kawaljit Singh, Kawaljit Singh et al. · European Journal of Medicinal Chemistry · 2011 · 76 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Antimalarial Pyrido[1,2-<i>a</i>]benzimidazoles: Lead Optimization, Parasite Life Cycle Stage Profile, Mechanistic Evaluation, Killing Kinetics, and in Vivo Oral Efficacy in a Mouse Model

Kawaljit Singh, John Okombo, Christel Brunschwig et al. · Journal of Medicinal Chemistry · 2017 · 45 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Antimalarial Pyrido[1,2-<i>a</i>]benzimidazole Derivatives with Mannich Base Side Chains: Synthesis, Pharmacological Evaluation, and Reactive Metabolite Trapping Studies

John Okombo, Christel Brunschwig, Kawaljit Singh et al. · ACS Infectious Diseases · 2019 · 39 citations

Medicine, Medicinal Chemistry, Pharmacology +17

Spiropyrimidinetrione DNA Gyrase Inhibitors with Potent and Selective Antituberculosis Activity

Preshendren Govender, Rudolf Müller, Kawaljit Singh et al. · Journal of Medicinal Chemistry · 2022 · 35 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Synthesis of new verapamil analogues and their evaluation in combination with rifampicin against Mycobacterium tuberculosis and molecular docking studies in the binding site of efflux protein Rv1258c

Kawaljit Singh, Malkeet Kumar, Elumalai Pavadai et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 34 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17